Die Struktur von Tadalafil erlaubt eine selektive Bindung an die Bindungsstelle der PDE5 und minimiert gleichzeitig die Interaktion mit PDE6, was visuelle Nebenwirkungen einschränkt. Seine Verteilung im Organismus erfolgt breit, wobei das Verteilungsvolumen etwa 63 Liter beträgt. Über 90 % des Wirkstoffs sind an Plasmaproteine gebunden. Die Wirkung bleibt unabhängig von der Nahrungsaufnahme konstant. Der Abbauweg über CYP3A4 kann durch Hemmer wie Ritonavir oder Ketoconazol verlangsamt werden, was die Plasmakonzentrationen deutlich erhöht. In diesem Kontext wird cialis 20mg preis häufig in Bezug auf pharmakokinetische Wechselwirkungen erwähnt.

Distanceriding.org

American Endurance Ride Conference
Rule 13 Appendices
Please see the AERC Rules and Regulations (revised December 1, 2011) for complete information about AERC drug rule policy.
Appendix A. Prohibited Substances
Acepromazine. Atrovet,.Notensil,.PromAce®.
Benazeprilat,.Benazepril.and.MC-tab.Lotrel,.
Acetaminophen.(Paracetamol).Tylenol,.Tempra,.etc.
Carticaine.(see.articaine). Septocaine;.
Cathinone.(khat,.kat,.qat,.quat,.chat,.catha,.
Albuterol.(Salbutamol).Proventil,.Ventolin.
Deoxycorticosterone. Percortin,.DOCA,.
Aldosterone. Aldocortin,.Electrocortin.
Chloral.hydrate. Nactec,.Oridrate,.etc.
Desipramine. Norpromine,.Pertofrane.
Aminoglycosides. Gentocin,.Amiglyde,.Tobrex,.
Chlorpheniramine.Chlortriemton,.etc.
Dibucaine. Nupercainal,.Cinchocaine.
amikacin,.tobramycin,.neomycin,.spectinomycin Chlorpromazine.Thorazine,.Largactil.
Diclofenac. Surpass,.Voltaren,.Voltarol.
Butabarbital.(Secbutobarbitone). Butacaps,.
Butamben.(butyl.aminobenzoate). Butesin.
Cloxazolam.Enadel,.Sepazon,.Tolestan.
Articaine.Septocaine;.Ultracaine,.etc.
Azaperone. Stresnil,.Suicalm,.Fentaz.(with.
Droperidol.Inapsine,.Droleptan,.Innovar-Vet.
A. Prohibited Substances . . .
Fluphenazine.Prolixin,.Permitil,.Anatensol,.etc.
Enalapril.(metabolite.enaloprilat).Vasotec.
Methotrimeprazine.Levoprome,.Neurocil,.etc.
Ergotamine. Gynergen,.Cafergot,.etc.
Fosinopril,.metabolite,.Fosinoprilat.Monopril Levothyroxine. Eltroxin,.Synthroid,.Soloxine,.
Erythropoietin.(EPO).Epogen,.Procrit,.etc.
Estazolam.Domnamid,.Eurodin,.Nuctalon.
Gamma-oryzanol.(other.than.naturally.occurs.
in.equine.feeds.such.as.rice.bran/rice.bran.oil) Guaifenesin.(glycerol.guiacolate). Gecolate Ethylaminobenzoate.(Benzocaine). Semets,.etc.
Macrolides. Zithromax,.Biaxxin.(including.
erythromycin,.azithromycin,.clarithromycin) Magnesium.sulphate.administered.for.the.
purpose.of.and.at.the.levels.of.providing.
a.calming/tranquilizing.effect.Magnesium.
Hemoglobin.glutamers.Oxyglobin.Hemopure.
sulphate.administered.as.an.electrolyte.
Moexipril.(metabolite,.moexiprilat).Uniretic.
Hydrocortisone.(Cortisol). Cortef,.etc.
Nabumetone.Anthraxan,.Relafen,.Reliflex.
Ibuprofen.Motrin,.Advil,.Nurpin,.etc.
Mephobarbital.(Methylphenobarbital).Mebaral.
Nandrolone.Nandrolin,.Laurabolin,.Durabolin.
Flunitrazepam. Rohypnol,.Narcozep,.Darkene,.
Fluoroquinolones. Baytril,.Cipro,.Ciloxan,.A180 Ketamine. Ketalar,.Ketaset,.Vetalar.
(including.enrofloxacin,.ciprofloxacin,.
Ketazolam.Anxon,.Laftram,.Solatran,.Loftran.
A. Prohibited Substances . . .
Omeprozole.Gastroguard,.Ulcerguard,.Prilosec,.
Trandolapril.(and.metabolite,.trandolaprilat) Secobarbital.(Quinalbarbitone).Seconal.
Spirapril,.metabolite.Spiraprilat. Renomax.
Succinylcholine. Sucostrin,.Quelin,.etc.
Prochlorperazine.Darbazine,.Compazine.
Sulfonamides.and.Potentiated.Sulfonamides.
Tribrissen,.Septra,.TMS.(sulfamethazine,.
(including.procaine.penicillin.G,.sodium.or.
Pentaerythritol.tetranitrate. Duotrate.
Pyrithyldione. Hybersulfan,.Sonodor.
Yucca.other.than.as.a.feed.additive.for.the.
Quinapril,.metabolite.Quinaprilat. Accupril.
purpose.of.and.at.the.levels.of.ammonia.
Ramipril,.metabolite.Ramiprilat. Altace.
Phenylephrine.Isophrin,.Neo-Synephrine.
Appendix B. Categories of Prohibited Substances
1. Anti-inflammatory. drugs. (steroidal. and/or. non- 12.Hormonal.products.(natural.or.synthesized).ex- steroidal).or.other.substances.that.have.similar.phar- cept.for.progesterone.or.similar.acting.progestagens.
in.mares.only,.administered.for.the.purpose.of.con- 2.Antipsychotic,.anti-epilectic.and.antihypertensive.
25. Bronchodialators. and. products. used. for. the.
13.Pharmacological.substances.designed.and.mar- treatment.of.recurrent.airway.disease,.mucolytics.and.
3.Antidepressants.such.as.selective.serotonin.reup- keted.primarily.for.human.use.or.use.in.other.species.
take. inhibitors,. monoamine. oxidase. inhibitors. and.
and. for. which. alternative. and. generally. accepted.
4.Tranquilizers.and.sedatives.including.benzodiaz- 14.Hypersensitizing.or.desensitizing.agents.
30.Topical.agents,.including.ophthalmic,.otic,.der- mal.and.wound.ointments.or.liniments.that.contain.
7. Amphetamines. and. other. central. nervous. system.
stimulants.including.cocaine.and.related.psychotic.drugs 19.Proton.pump.inhibitors.and.H2.receptor.antago- 31. Any. substance. administered. while. competing.
in.an.endurance.ride.by.nasogastric.tube.or.syringe/ 10.Anabolic.steroids.and.growth.promoters 21.Substances.designed,.marketed,.and/or.admin- 32. Yucca. administered. for. the. purpose. of. and. at.
11.Peptides.and.genetically.recombinant.substanc- istered.to.affect.the.behavior.of.an.equine.in.a.calm- the.levels.of.ammonia.reduction.and.intestinal.health.
es.such.as.erythropoietin,.insulin.growth.factor.and.
ing.(tranquilizing).or.energizing.(stimulating).manner.
Yucca.administered.for.any.other.purpose.or.at.levels.
This.is.to.include.herbal.and/or.natural.products.
to.provide.anti-inflammatory.effect.is.prohibited.
Appendix C. Allowed Substances
1.Vitamins.(other.than.thiamine.administered.for.the.
7.Progesterone.and.similar.acting.progestagens.such.
purpose.of.providing.a.calming/tranquilizing.effect) as. altrenogest. (Regumate). only. in. mares. to. control.
12.Magnesium.sulphate.admistered.for.the.purpose.
8. The. fol owing. chondroprotective. agents:. glucos- of.electrolyte.supplementation.Magnesium.sulphate.
4. Topical.agents.such.as.liniments.and.wound.dressings.
amine,. chondroitin. sulfate,. polysulfated. glycosami- administered.for.the.purpose.of.and.at.the.levels.of.
that.do.not.contain.a.prohibited.substance noglycan,. hyaluronate. Not. to. be. administered. by.
providing.a.calming/tranquilizing.effect.is.prohibited.
needle/syringe.while.competing.in.an.endurance.ride.
6.Ice.and.ice.water.administered.orally.and/or.topi- *There.is.insufficient.information.available.to.advise.
9. Acid. neutralizers. including. aluminum. hydroxide.
as.to.the.timing.of.administration.close.to.the.time.
Appendix D. Threshhold Levels
Urinary.thresholds.refer.to.the.parent.drug.and/or.metabolite.S.=.stallions,.G.=.geldings,.M.=.mares) Flunixin.(Banamine). 50.ng/ml. plasma.
. (epitestosterone). 20.ng/ml.(G). urine.
*The.threshold.for.furosemide.applies.only.if.the.urine.
Dimethylsulfoxide.(DMSO). 15,000.ng/ml. urine specific.gravity.is.less.than.1.010.
Appendix E. Known Detection Times for Substances Used Therapeutically in the Horse
Typical Dose/Route* for
Elimination Detection Limit
Drug (Brand Name)
Therapeutic Indication
1000 lb. (450kg) Horse
Half-Life
Source of Info.
____________________________________________________________________________________________________________________________________________________________
Tranquilizers/Sedatives
____________________________________________________________________________________________________________________________________________________________acepromazine.(Atravet®,.PromAce®).
Tranquilizer.used.for.calming.horses. Has.no.pain-relieving.action.
____________________________________________________________________________________________________________________________________________________________butorphanol.(Torbugesic®).
Sedative.with.pain-relieving.action,.used.frequently.to.treat.colic.in.horses.
____________________________________________________________________________________________________________________________________________________________dantrolene.(Dantrium®).
Muscle.relaxant.used.in.horses.with.myopathies.(“tying-up”).
____________________________________________________________________________________________________________________________________________________________detomidine.(Dormosedan®).
Sedative.with.pain-relieving.action,.used.frequently.to.treat.colic.in.horses.
____________________________________________________________________________________________________________________________________________________________guaifenesin.(Guailaxin®,.Gecolate®).
Muscle.relaxant.used.in.horses.with.myopathies.(“tying-up”).
____________________________________________________________________________________________________________________________________________________________methocarbamol.(Robaxin®).
Muscle.relaxant.used.in.horses.with.myopathies.(“tying-up”).
____________________________________________________________________________________________________________________________________________________________romifidine.(Sedivet®).
Sedative.with.pain-relieving.action,.used.frequently.to.treat.colic.in.horses.
____________________________________________________________________________________________________________________________________________________________
Anti-inflammatories/Pain Relievers
____________________________________________________________________________________________________________________________________________________________aspirin.
Oral y.or.pain-reliever.in.the.horse. Sometimes.used.to.treat.periodic.ophthalmia. 11.7.grams.Orally.
(“moon.blindness”),.laminitis,.and.colic.due.to.parasite.damage.
____________________________________________________________________________________________________________________________________________________________diclofenac.sodium.(Surpass).
Applied.topically.as.an.anti-inflammatory.agent.
Five-inch.ribbon.of.1%.cream. N/A**.
____________________________________________________________________________________________________________________________________________________________dimethylsulfoxide.(DMSO).
Applied.topically.as.an.anti-inflammatory.agent,.given.IV.to.treat.myopathies. 19.8.grams.topically.
____________________________________________________________________________________________________________________________________________________________flunixin.meglumine.(Banamine®).
Nonsteroidal.anti-inflammatory.drug.used.to.treat.colic.and.
musculoskeletal.pain.and.inflammation.
____________________________________________________________________________________________________________________________________________________________ketoprofen.(Ketofen®,.Anafen®).
Nonsteroidal.anti-inflammatory.drug.used.to.treat.colic.
and.musculoskeletal.pain.and.inflammation.
____________________________________________________________________________________________________________________________________________________________lidocaine.(Xylocaine®).
Local.anesthetic.used.to.block.nerves.
____________________________________________________________________________________________________________________________________________________________meclofenamic.acid.(Arquel®).
Nonsteroidal.anti-inflammatory.drug.used.to.treat.colic.and.
musculoskeletal.pain.and.inflammation.
____________________________________________________________________________________________________________________________________________________________mepivicaine.(Carbocaine®).
Local.anesthetic.used.to.block.nerves.
____________________________________________________________________________________________________________________________________________________________naproxen.(Equiproxen,.Aleeve®).
Nonsteroidal.anti-inflammatory.drug.used.to.treat.colic.and.
musculoskeletal.pain.and.inflammation.
____________________________________________________________________________________________________________________________________________________________pergolide.(Permax,.Teva).
____________________________________________________________________________________________________________________________________________________________phenylbutazone.(“Bute”).
Nonsteroidal.anti-inflammatory.drug.used.to.treat.colic.and.
musculoskeletal.pain.and.inflammation.
____________________________________________________________________________________________________________________________________________________________procaine.(Novocaine®).
Local.anesthetic.used.to.block.nerves.
____________________________________________________________________________________________________________________________________________________________procaine.penicillin.G.
Combined.with.penicillin.to.make.the.antibiotic.slowly.absorbed.from.the.
injection.site,.to.give.it.a.long.duration.of.antibacterial.action.
____________________________________________________________________________________________________________________________________________________________
Corticosteroids
____________________________________________________________________________________________________________________________________________________________betamethasone.(Betasone®,.Celestone®). Anti-inflammatory;.allergic.reactions.
____________________________________________________________________________________________________________________________________________________________dexamethasone.(Azium®).
Anti-inflammatory;.allergic.reactions.
____________________________________________________________________________________________________________________________________________________________flumethasone.(Flucort®).
Anti-inflammatory;.allergic.reactions.
____________________________________________________________________________________________________________________________________________________________isoflupredone.(Predef.2X®).
Anti-inflammatory;.allergic.reactions.
____________________________________________________________________________________________________________________________________________________________methylprednisolone.acetate.
Anti-inflammatory;.allergic.reactions.
____________________________________________________________________________________________________________________________________________________________prednisolone.
Anti-inflammatory;.allergic.reactions.
____________________________________________________________________________________________________________________________________________________________prednisone.
Anti-inflammatory;.allergic.reactions.
____________________________________________________________________________________________________________________________________________________________triamcinolone.(Vetalog®).
Anti-inflammatory;.allergic.reactions.
____________________________________________________________________________________________________________________________________________________________
Miscellaneous Drugs
____________________________________________________________________________________________________________________________________________________________aminophylline.
Opens.airways.in.horses.with.“heaves”.
____________________________________________________________________________________________________________________________________________________________clenbuterol.(Ventipulmin®).
Opens.airways.in.horses.with.“heaves”.
____________________________________________________________________________________________________________________________________________________________dembrexine.(Sputolysin®).
Expectorant.for.horses.with.“heaves”.
____________________________________________________________________________________________________________________________________________________________diphenhydramine.(Benadryl®).
____________________________________________________________________________________________________________________________________________________________isoxuprine.(Vasodilan®).
Dilates.blood.vessels,.used.for.treatment.of.navicular.disease.
____________________________________________________________________________________________________________________________________________________________omeprazole.(Gastrogard®,.Ulcergard®). Proton.pum.inhibitor.used.for.the.treatment.of.esophagitis,.erosive.
____________________________________________________________________________________________________________________________________________________________theophylline.
Opens.airways.in.horses.with.“heaves”.
____________________________________________________________________________________________________________________________________________________________*.IV.-.intravenous,.IM.-.Intramuscular,.SC.-.Subcutaneous,.IA.-.Intra-articular.(into.the.joint);. **.No.information.available.
Appendix F. Prohibited Treatments
1.Acupuncture,.or.any.procedure.involving.the.
Appendix.G.item.4).for.the.purpose.of.administer- points. This.would.include.but.not.be.limited.to.
insertion.of.a.needle.into.the.equine.
ing.a.substance.or.to.stimulate.a.response.
2.Osseous.manipulation.(chiropractic).
5.Extracorporeal.Shockwave.therapy.or.similar.
7.Administration.of.a.local.anesthetic,.either.
3. Any. manipulative. procedure. using. an. ex- device. to. produce. a. temporary. or. permanent.
topical,.injectable.or.oral.to.any.part.of.the.horse.
ternal.device.or.instrument.such.as.devices.to.
analgesia.This.would.also.include.radiofrequency.
or.any.procedure.that.results.in.desensitization.
manipulate.or.stimulate.acupressure.or.response.
(RF). neurectomy. Extracorporeal. shockwave.
points,.including.but.not.limited.to.bioscans,.laser.
therapy.is.not.permitted.within.7.days.of.com- 8.Pinfiring/pinfreezing.–.visible.active,.open.
lesions.from.such.a.procedure.would.prohibit.a.
4.Any.procedure.involving.the.placement.of.a.
6. Any. external. magnetic. field. device. or.
tube.or.other.instrument.into.the.equine.(other.
electropulse. generator. device. applied. either.
9.The.use.of.substances.or.devices.that.cool.
than.the.oral.cavity.using.a.dosing.syringe,.see.
over.the.entire.body.or.specifically.on.pressure.
Appendix G. Allowable Treatments
1.Massage,.deep.massage/acupressure.using.digital.(hand/finger).pres- ice. water. The. use. of. devices. or. substances. that. cool. below. 0. degrees.
2.The.use.of.instruments.commonly.know.as.grooming.instruments.
4.The.oral.administration.of.permitted.substances.by.means.of.dosing.
3.The.use.of.ice.boots.and.other.means.of.applying.ice/ice.water.topical y.
Can.include.the.use.of.compression.wraps.as.well.as.devices.that.circulate.
5.Healed.scars.from.pinfiring.are.allowed.

Source: http://www.distanceriding.org/php/articles/vets/DrugRuleAppendices-2011.pdf

rose.ofai.at

Does Irrelevant Information Play a Role in Judgment? Boicho Kokinov ([email protected])12 Penka Hristova ([email protected])1 Georgi Petkov ([email protected])1 1Central and East European Center for Cognitive Science, Department of Cognitive Science and Psychology,New Bulgarian University, 21 Montevideo Street2Institute of Mathematics and Informatics, Bulgarian Academy of Science

Pii: s0090-4295(02)01903-9

PEDIATRIC UROLOGY PROSPECTIVE COMPARISON AND 1-YEAR FOLLOW-UP OFDEXTRANOMER/HYALURONIC ACID COPOLYMER INJECTIONFOR TREATMENT OF VESICOURETERAL REFLUX IN CHILDRENJ. OSWALD, M. RICCABONA, L. LUSUARDI, G. BARTSCH, AND C. RADMAYR ABSTRACT Objectives. To compare, in a prospective study, the efficacy of a single injection of polydimethylsiloxane (Macroplastique) or dextranomer/hyaluronic ac

Copyright © 2010-2014 Medical Articles